856243-80-6

Degrasyn Chemical Structure
856243-80-6

Chemical Structure

Degrasyn

Synonym(s): WP1130

  • CAS No.: 856243-80-6
  • Formula:C19H18BrN3O
  • Molecular Weight:384.27

IUPAC Name: (S,E)-3-(6-bromopyridin-2-yl)-2-cyano-N-(1-phenylbutyl)acrylamide

InChIKey: LIDOPKHSVQTSJY-VMEIHUARSA-N

SMILES: BrC1=CC=CC(/C=C(C(N[C@H](C2=CC=CC=C2)CCC)=O)\C#N)=N1

Biological Activity: Degrasyn (WP1130) is a cell-permeable deubiquitinase (DUB) inhibitor, directly inhibiting DUB activity of USP9x, USP5, USP14, and UCH37. Degrasyn has been shown to downregulate the antiapoptotic proteins Bcr-Abl and JAK2.

Cat. No. Product Name Purity Description Pricing
HY-13264 		Degrasyn 99.70% Degrasyn (WP1130) is a cell-permeable deubiquitinase (DUB) inhibitor, directly inhibiting DUB activity of USP9x, USP5, USP14, and UCH37. Degrasyn has been shown to downregulate the antiapoptotic proteins Bcr-Abl and JAK2.
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This product is a controlled substance and not for sale in your territory.

This product is not for sale in your territory.

This compound is listed in the SVHC (Substances of Very High Concern) candidate list of ECHA (European Chemicals Agency).

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