GEMSA
GEMSA is a potent inhibitor of enkephalin convertase (Ki=8.8 nM). GEMSA elicites analgesia.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- Reinheit : 98%
- CAS. Nr.: 77482-44-1
- Formel: C7H13N3O4S
- Molecular Weight:235.26
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Speicherung:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
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Biologische Aktivität
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Chemical Information
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Help & FAQs
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HY-100788
2-PMPAGCPII Inhibitor -
HY-103345
2-MPPAGCP II Inhibitor -
HY-100788R
2-PMPA (Standard)Standard -
HY-103345R
2-MPPA (Standard)GCP II Inhibitor -
HY-103344
ZJ43NAAG Peptidase Inhibitor -
HY-W704574
MergetpaCarboxypeptidase Inhibitor -
HY-W044764
2-Benzylsuccinic acidCPA Inhibitor -
HY-70005
CPA inhibitorCPA Inhibitor -
HY-70003
Carboxypeptidase G2 (CPG2) InhibitorCPG2 Inhibitor -
HY-139840A
GCPII-IN-1 TFAGCPII Inhibitor -
HY-W044764R
2-Benzylsuccinic acid (Standard)CPA Inhibitor
Biologische Aktivität
Beschreibung
IC50 & Target
Encephalin convertase, Ki 值为8.8 nM.
In Vitro
GEMSA inhibits the activation of TAFI and porcine CBB[1]. GEMSA can inhibit the prolongation of lysis time in recombinant BAP and does not lead to the lysis of APC fibronectin[1]. GEMSA inhibits the prolongation of lysis time in porcine CPB, TAFI, and recombinant BAP, APC with the EC50 values of 0.34 μM, 100μM, 115 μM, 90 μM respectively[1][2].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. .
In Vivo
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS. Nr. 77482-44-1
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Appearance Solid
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Molecular Weight 235.26
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Formel C7H13N3O4S
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Color White to off-white
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SMILES
OC(C(SCCNC(N)=N)CC(O)=O)=O
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Synonyms
2-Guanidinoethylmercaptosuccinic acid
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Reinheit & Dokumentation
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Data Sheet (266 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
GEMSA Related Classifications
HY-118120 Related Classifications
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