(R)-PAD-PF2
Based on 1 Customer Validation
(R)-PAD-PF2 is an isomer of PAD-PF2 (HY-176710). PAD-PF2 is a PAD family inhibitor, as well as a κ-opioid receptor agonist (EC50 = 7.55 μM) and an M1 muscarinic acetylcholine receptor antagonist (IC50 = 12.3 μM).
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- Reinheit: 99.95%
- Formel: C25H27Cl2N5O
- Molecular Weight:484.42
-
Speicherung:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
Biologische Aktivität
Chemical Information
-
Appearance Solid
-
Molecular Weight 484.42
-
Formel C25H27Cl2N5O
-
Color White to off-white
-
SMILES
O=C(N1CCCC1)[C@H](N)C2CCN(C3=NC=CC4=C3C=CC=C4C5=NC=C(Cl)C=C5Cl)CC2
-
Versand
Room temperature in continental US; may vary elsewhere.
-
Speicherung
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Lösungsmittel & Löslichkeit
DMSO : 100 mg/mL (206.43 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
Reinheit & Dokumentation
-
Data Sheet (242 KB)
-
SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
-
Handling Instructions (2659 KB)
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.0643 mL | 10.3216 mL | 20.6432 mL | 51.6081 mL |
| 5 mM | 0.4129 mL | 2.0643 mL | 4.1286 mL | 10.3216 mL | |
| 10 mM | 0.2064 mL | 1.0322 mL | 2.0643 mL | 5.1608 mL | |
| 15 mM | 0.1376 mL | 0.6881 mL | 1.3762 mL | 3.4405 mL | |
| 20 mM | 0.1032 mL | 0.5161 mL | 1.0322 mL | 2.5804 mL | |
| 25 mM | 0.0826 mL | 0.4129 mL | 0.8257 mL | 2.0643 mL | |
| 30 mM | 0.0688 mL | 0.3441 mL | 0.6881 mL | 1.7203 mL | |
| 40 mM | 0.0516 mL | 0.2580 mL | 0.5161 mL | 1.2902 mL | |
| 50 mM | 0.0413 mL | 0.2064 mL | 0.4129 mL | 1.0322 mL | |
| 60 mM | 0.0344 mL | 0.1720 mL | 0.3441 mL | 0.8601 mL | |
| 80 mM | 0.0258 mL | 0.1290 mL | 0.2580 mL | 0.6451 mL | |
| 100 mM | 0.0206 mL | 0.1032 mL | 0.2064 mL | 0.5161 mL |