CB1-IN-2
CB1-IN-2 (Compound 4g) is a selective CB1 inhibitor with an IC50 of 0.644 μM. CB1-IN-2 can penetrates BBB and might cause CNS side effect similar with Rimonabant.
For research use only. We do not sell to patients.
- CAS No.: 2527805-39-4
- Formula: C17H19Cl2N5O
- Molecular Weight:380.27
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Description
IC50 & Target
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CB1 0.644 μM (IC50) |
Chemical Information
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CAS No. 2527805-39-4
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Molecular Weight 380.27
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Formula C17H19Cl2N5O
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SMILES
O=C(C1=NN(C2=CC=C(Cl)C=C2Cl)C(C3CC3)=N1)NN4CCCCC4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Protocols
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Cell Cytotoxicity Assay
Cytotoxicity assays are usually based on the assessment of cell membrane damage, which can also be indirectly detected by measuring cell viability. Detection methods include MTT assay, CKK-8 assay, LDH assay and ATP assay, etc.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)