VU6036864
VU6036864 (compound 45) is an orally active, selective mAChR M5 antagonist with IC50=20 nM for human M5. VU6036864 is >500-fold selective for human M1-4, with BBB characteristic and high oral bioavailability (%F>100%).
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- CAS No.: 2746406-36-8
- Formule: C15H12D4ClN5O3S
- Masse moléculaire:385.86
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
IC50: 20 nM (human mAChR M5)[1]
1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.
Chemical Information
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CAS No. 2746406-36-8
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Unlabeled Cas 2746405-41-2
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Masse moléculaire 385.86
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Formule C15H12D4ClN5O3S
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SMILES
CC1=NC=C(S(=O)(N2C([2H])([2H])CC(C3=CN4C(C=C3Cl)=NC=N4)CC2([2H])[2H])=O)O1
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
VU6036864 Related Classifications
HY-159578S Related Classifications
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