CXCR4-IN-2
CXCR4-IN-2 (compound A1) is a bifunctional fluorinated small molecule that is a potent CXCR4 inhibitor with anticancer activity. CXCR4-IN-2 has cytotoxic (IC50: 60 μg/mL; 72 h) and antiproliferative effects on mouse colorectal cancer (CRC) cells. CXCR4-IN-2 induces cell arrest in the G2/M phase and induces apoptosis.
For research use only. We do not sell to patients.
- Formula: C21H20F6N4S
- Molecular Weight:474.47
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Chemical Information
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Molecular Weight 474.47
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Formula C21H20F6N4S
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SMILES
CC1=CC=C(/N=C(NC(N/C(C(F)(F)F)=N/C2=CC(C)=C(C)C=C2)=S)\C(F)(F)F)C=C1C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)