Debrisoquin hemisulfate
Based on 1 Customer Validation
Debrisoquin (Isocaramidine) hemisulfate is a TMPRSS2 inhibitors that inhibits SARS-CoV-2 entry into human lung cell line by a TMPRSS2-depedent manner, with an IC50 of 22μM. Debrisoquin hemisulfate can be used for antiviral research.
For research use only. We do not sell to patients.
- Purity: 99.9%
- CAS No.: 581-88-4
- Formula: C10H13N3.1/2H2O4S
- Molecular Weight:224.27
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Storage:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
All Endogenous Metabolite Isoforms
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Biological Activity
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Human Endogenous Metabolite |
Chemical Information
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CAS No. 581-88-4
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Appearance Solid
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Molecular Weight 224.27
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Formula C10H13N3.1/2H2O4S
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Color Light yellow to yellow
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SMILES
O=S(O)(O)=O.N=C(N1CC2=C(CC1)C=CC=C2)N.[1/2]
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Synonyms
Debrisoquine hemisulfate; Isocaramidine hemisulfate; Ro 5-3307/1 hemisulfate
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Structure Classification
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Initial Source
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
H2O : 10.42 mg/mL (46.46 mM; ultrasonic and warming and heat to 60°C)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (240 KB)
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SDS (392 KB)
- English - EN (392 KB)
- Français - FR (392 KB)
- Deutsch - DE (392 KB)
- Norwegian - NO (392 KB)
- Español - ES (392 KB)
- Swedish - SV (392 KB)
- Italian - IT (392 KB)
- Korean - KR (392 KB)
- Portuguese - PT (392 KB)
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Handling Instructions (2659 KB)
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| H2O | 1 mM | 4.4589 mL | 22.2946 mL | 44.5891 mL | 111.4728 mL |
| 5 mM | 0.8918 mL | 4.4589 mL | 8.9178 mL | 22.2946 mL | |
| 10 mM | 0.4459 mL | 2.2295 mL | 4.4589 mL | 11.1473 mL | |
| 15 mM | 0.2973 mL | 1.4863 mL | 2.9726 mL | 7.4315 mL | |
| 20 mM | 0.2229 mL | 1.1147 mL | 2.2295 mL | 5.5736 mL | |
| 25 mM | 0.1784 mL | 0.8918 mL | 1.7836 mL | 4.4589 mL | |
| 30 mM | 0.1486 mL | 0.7432 mL | 1.4863 mL | 3.7158 mL | |
| 40 mM | 0.1115 mL | 0.5574 mL | 1.1147 mL | 2.7868 mL |
* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.