Debrisoquin hydroiodide
Based on 1 Customer Validation
Debrisoquin (hydroiodide) is the hydrochloride form of Debrisoquin (HY-B1624). Debrisoquin is a TMPRSS2 inhibitors that inhibits SARS-CoV-2 entry into human lung cell line by a TMPRSS2-depedent manner. Debrisoquin can be used for antiviral research.
For research use only. We do not sell to patients.
- Purity: 99.84%
- CAS No.: 1052540-65-4
- Formula: C10H14IN3
- Molecular Weight:303.14
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Storage:
4°C, protect from light
* In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
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Solvent & Solubility
- Purity & Documentation
- References
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Help & FAQs
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Biological Activity
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 1052540-65-4
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Appearance Solid
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Molecular Weight 303.14
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Formula C10H14IN3
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Color Off-white to light yellow
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SMILES
N=C(N1CC2=C(CC1)C=CC=C2)N.I
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Synonyms
Debrisoquine hydroiodide; Isocaramidine hydroiodide; Ro 5-3307/1 hydroiodide
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
4°C, protect from light
* In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
Solvent & Solubility
DMSO : 175 mg/mL (577.29 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
H2O : 25 mg/mL (82.47 mM; ultrasonic and warming and heat to 60°C)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (270 KB)
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SDS (394 KB)
- English - EN (394 KB)
- Français - FR (394 KB)
- Deutsch - DE (394 KB)
- Norwegian - NO (394 KB)
- Español - ES (394 KB)
- Swedish - SV (394 KB)
- Italian - IT (394 KB)
- Korean - KR (394 KB)
- Portuguese - PT (394 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| H2O / DMSO | 1 mM | 3.2988 mL | 16.4940 mL | 32.9881 mL | 82.4701 mL |
| 5 mM | 0.6598 mL | 3.2988 mL | 6.5976 mL | 16.4940 mL | |
| 10 mM | 0.3299 mL | 1.6494 mL | 3.2988 mL | 8.2470 mL | |
| 15 mM | 0.2199 mL | 1.0996 mL | 2.1992 mL | 5.4980 mL | |
| 20 mM | 0.1649 mL | 0.8247 mL | 1.6494 mL | 4.1235 mL | |
| 25 mM | 0.1320 mL | 0.6598 mL | 1.3195 mL | 3.2988 mL | |
| 30 mM | 0.1100 mL | 0.5498 mL | 1.0996 mL | 2.7490 mL | |
| 40 mM | 0.0825 mL | 0.4124 mL | 0.8247 mL | 2.0618 mL | |
| 50 mM | 0.0660 mL | 0.3299 mL | 0.6598 mL | 1.6494 mL | |
| 60 mM | 0.0550 mL | 0.2749 mL | 0.5498 mL | 1.3745 mL | |
| 80 mM | 0.0412 mL | 0.2062 mL | 0.4124 mL | 1.0309 mL | |
| DMSO | 100 mM | 0.0330 mL | 0.1649 mL | 0.3299 mL | 0.8247 mL |
* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.
Debrisoquin hydroiodide Related Classifications
HY-W195509 Related Classifications
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