1. GPCR/G Protein Neuronal Signaling
  2. 5-HT Receptor
  3. Dehydroaripiprazole hydrochloride

Dehydroaripiprazole hydrochloride  (Synonyms: OPC-14857 hydrochloride; DM-14857 hydrochloride)

Cat. No.: HY-113575
Handling Instructions

Dehydroaripiprazole (OPC-14857) hydrochloride is an active metabolite of Aripiprazole. Aripiprazole is an antipsychotic agent and is metabolized by CYP3A4 and CYP2D6 forming mainly Dehydroaripiprazole hydrochloride. Dehydroaripiprazole hydrochloride has with antipsychotic activity equivalent to Aripiprazole.

For research use only. We do not sell to patients.

Dehydroaripiprazole hydrochloride Chemical Structure

Dehydroaripiprazole hydrochloride Chemical Structure

CAS No. : 1008531-60-9

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Description

Dehydroaripiprazole (OPC-14857) hydrochloride is an active metabolite of Aripiprazole. Aripiprazole is an antipsychotic agent and is metabolized by CYP3A4 and CYP2D6 forming mainly Dehydroaripiprazole hydrochloride. Dehydroaripiprazole hydrochloride has with antipsychotic activity equivalent to Aripiprazole[1][2][3][4].

IC50 & Target[4]

5-HT1A Receptor

4.2 nM (Ki)

Molecular Weight

482.83

Formula

C23H26Cl3N3O2

CAS No.
SMILES

O=C1NC2=C(C=CC(OCCCCN3CCN(C4=CC=CC(Cl)=C4Cl)CC3)=C2)C=C1.Cl

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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Dehydroaripiprazole hydrochloride Related Classifications

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
Dehydroaripiprazole hydrochloride
Cat. No.:
HY-113575
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