1. GPCR/G Protein
    Neuronal Signaling
  2. 5-HT Receptor
  3. Dehydroaripiprazole

Dehydroaripiprazole (Synonyms: OPC-14857; DM-14857)

Cat. No.: HY-100665
Handling Instructions

Dehydroaripiprazole (OPC-14857) is an active metabolite of Aripiprazole. Aripiprazole is an antipsychotic agent and is metabolized by CYP3A4 and CYP2D6 forming mainly Dehydroaripiprazole. Dehydroaripiprazole has with antipsychotic activity equivalent to Aripiprazole.

For research use only. We do not sell to patients.

Dehydroaripiprazole Chemical Structure

Dehydroaripiprazole Chemical Structure

CAS No. : 129722-25-4

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Description

Dehydroaripiprazole (OPC-14857) is an active metabolite of Aripiprazole. Aripiprazole is an antipsychotic agent and is metabolized by CYP3A4 and CYP2D6 forming mainly Dehydroaripiprazole. Dehydroaripiprazole has with antipsychotic activity equivalent to Aripiprazole[1][2][3].

IC50 & Target[4]

5-HT1A Receptor

4.2 nM (Ki)

Molecular Weight

446.37

Formula

C₂₃H₂₅Cl₂N₃O₂

CAS No.

129722-25-4

SMILES

O=C1NC2=C(C=CC(OCCCCN3CCN(C4=CC=CC(Cl)=C4Cl)CC3)=C2)C=C1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

DehydroaripiprazoleOPC-14857 DM-14857OPC14857OPC 14857DM14857DM 14857DM-148575-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorMetaboliteCYP3A4CYP2D6antipsychoticInhibitorinhibitorinhibit

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Dehydroaripiprazole
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