ecMetAP-IN-1
Based on 1 Customer Validation
ecMetAP-IN-1 is an inhibitor of E. coli methionine aminopeptidase (ecMetAP) with an IC50 of 2.086 μM. ecMetAP-IN-1 is applicable to research related to bacterial infections caused by E. coli.
For research use only. We do not sell to patients.
- Purity: 98.12%
- CAS No.: 7471-12-7
- Formula: C13H11N3
- Molecular Weight:209.25
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Storage:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
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Solvent & Solubility
- Purity & Documentation
- References
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Help & FAQs
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Bioactive Compound Library Max
HY-L181
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Bioactive Compound Library
HY-L001
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Anti-Infection Compound Library
HY-L002
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Metabolism/Protease Compound Library
HY-L012
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Antibacterial Compound Library
HY-L049
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Metabolic Enzyme Compound Library
HY-L146
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MCE Bioactive Compound Library
HY-L001V
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High-Throughput Bioactive Compound Library
HY-L205
Biological Activity
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| Sf9 | IC50 |
7.7 μM
Compound: 16
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Inhibition of human MetAP2 expressed in baculovirus infected Sf9 cells
Inhibition of human MetAP2 expressed in baculovirus infected Sf9 cells
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[PMID: 20621724] |
ecMetAP-IN-1 (Compound 17) (45 min) inhibits CoII-Loaded Escherichia coli methionine aminopeptidase with an IC50 value of 2.086 μM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 7471-12-7
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Appearance Solid
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Molecular Weight 209.25
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Formula C13H11N3
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Color White to off-white
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SMILES
CC1=CC=C2N=C(C3=NC=CC=C3)NC2=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : 100 mg/mL (477.90 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (270 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 4.7790 mL | 23.8949 mL | 47.7897 mL | 119.4743 mL |
| 5 mM | 0.9558 mL | 4.7790 mL | 9.5579 mL | 23.8949 mL | |
| 10 mM | 0.4779 mL | 2.3895 mL | 4.7790 mL | 11.9474 mL | |
| 15 mM | 0.3186 mL | 1.5930 mL | 3.1860 mL | 7.9650 mL | |
| 20 mM | 0.2389 mL | 1.1947 mL | 2.3895 mL | 5.9737 mL | |
| 25 mM | 0.1912 mL | 0.9558 mL | 1.9116 mL | 4.7790 mL | |
| 30 mM | 0.1593 mL | 0.7965 mL | 1.5930 mL | 3.9825 mL | |
| 40 mM | 0.1195 mL | 0.5974 mL | 1.1947 mL | 2.9869 mL | |
| 50 mM | 0.0956 mL | 0.4779 mL | 0.9558 mL | 2.3895 mL | |
| 60 mM | 0.0796 mL | 0.3982 mL | 0.7965 mL | 1.9912 mL | |
| 80 mM | 0.0597 mL | 0.2987 mL | 0.5974 mL | 1.4934 mL | |
| 100 mM | 0.0478 mL | 0.2389 mL | 0.4779 mL | 1.1947 mL |
ecMetAP-IN-1 Related Classifications
HY-148442 Related Classifications
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