Enpatoran (Standard)

(Synonyms: M5049 (Standard))

Enpatoran (Standard) is the analytical standard of Enpatoran (HY-134581). This product is intended for research and analytical applications. Enpatoran (M5049) is a potent, orally active and dual TLR7/8 inhibitor with IC50s of 11.1 nM and 24.1 nM in HEK293 cells, respectively. Enpatoran is inactive against TLR3, TLR4 and TLR9. Enpatoran can block molecule synthetic ligands and natural endogenous RNA ligands. Enpatoran exhibits excellent pharmacoKinetic properties in vivo. Enpatoran can be used for both innate and adaptive autoimmunity blocKing research .

For research use only. We do not sell to patients.

  • CAS No.: 2101938-42-3
  • Formula: C16H15F3N4
  • Molecular Weight:320.31
  • Storage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

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100 mg

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