EP300/CBP ligand 3
CBP/p300 ligand 11 is a ligand of EP300 and CBP, which can be used for PROTAC synthesis, such as serving as the target protein ligand of PROTAC CBP/EP300 Degrader-5 (HY-184453).
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- Formule: C27H28N4O3
- Masse moléculaire:456.54
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
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EP300 |
CBP |
CBP/p300 ligand 11 is the target protein ligand of PROTAC CBP/EP300 Degrader-5 (HY-184453). PROTAC CBP/EP300 Degrader-5 is a PROTAC degrader targeting CBP and EP300, which induces G1-phase cell cycle arrest and triggers apoptosis. PROTAC CBP/EP300 Degrader-5 can be used in research related to EP300-dependent malignancies[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Masse moléculaire 456.54
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Formule C27H28N4O3
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SMILES
O=C([C@@H]1N(C(C2(C3=CC=C(OCC#C)C=C3)CCCC2)=O)CCC1)NC4=CC=CC5=C4C=NN5
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)