HJP 272
HJP 272 is a selective endothelin peptide A (ETA) receptor antagonist with an IC50 of 37.01 nM. . HJP 272 can be used for the researches of pulmonary arterial hypertension, fibrosis, renal failure and cancer.
For research use only. We do not sell to patients.
- CAS No.: 1072467-37-8
- Formula: C28H23NO8
- Molecular Weight:501.48
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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ETA 37.01 nM (IC50) |
ETB 15602.3 nM (IC50) |
HJP 272 (Compound 41) acts as an ETA-selective receptor antagonist in HEK293T cells, with an ETA IC50 of 37.01 nM and 421-fold selectivity over the ETB receptor[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 1072467-37-8
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Molecular Weight 501.48
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Formula C28H23NO8
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SMILES
O=C(C1=CC=CC(CC2=C(C(O)=O)N(CC3=CC4=C(C=C3CC)OCO4)C5=CC=C(O)C=C5C2=O)=C1)O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
HJP 272 Related Classifications
HY-183141 Related Classifications
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