FGH31
FGH31 (Compound 24) is a potent, selective, GRK2 dependency dopamine D4 agonist, with the Ki of 1.6 nM. FGH31 partial activates β- arrestin.
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- No. CAS: 3033813-47-4
- Fòrmula: C33H36N4O2
- Peso molecular:520.66
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Ver todos los productos específicos de isoformas Dopamine Receptor
MoreVer todos los productos específicos de isoformas Arrestin
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Actividad biológica
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Dopamine D4 receptor 1.6 nM (Ki) |
GRK2 |
FGH31 (Compound 24) (50 μM) decreases at a similar rate as Imipramine (HY-B1490A) in rat liver microsomes[1].
FGH31 (50 μM, 4 h) shows no significant transport by P-glycoprotein (P-gp) in Caco-2 cells[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 3033813-47-4
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Peso molecular 520.66
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Fòrmula C33H36N4O2
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SMILES
O=C(NCCCN1CCN(C2=CC=CC=C2OC)CC1)NC3=CC=CC=C3C4=CC=C(C5=CC=CC=C5)C=C4
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
FGH31 Related Classifications
HY-155099 Related Classifications
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