M4K2163
M4K2163 is a ALK2 inhibitor that serves as a target protein ligand for the synthesis of PROTACs, such as M4K3250 (HY-183718). M4K2163 induces cytotoxic effects in glioblastoma cells. M4K2163 can be used in the research of diffuse intrinsic pontine glioma and glioblastoma.
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- No. CAS: 2600795-21-7
- Fòrmula: C24H26FN3O2
- Peso molecular:407.48
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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Chemical Information
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Actividad biológica
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ALK2 |
M4K2163 (96 h) reduces viability of U87-MG glioblastoma cells in a dose-dependent manner over 96 h, with cytotoxic activity independent of CRBN recruitment[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 2600795-21-7
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Peso molecular 407.48
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Fòrmula C24H26FN3O2
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SMILES
CC1=C(C2=CC=C(N3CCNCC3)C=C2)C=NC=C1C4=CC(OC)=C(F)C(OC)=C4
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
M4K2163 Related Classifications
HY-183720 Related Classifications
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