MDA7
MDA7 is the selective agonist for cannabinoid receptor 2 with EC50 of 128 nM and 67.4 nM in human CB2 receptor and rat CB2 receptor. MDA7 exhibits good affinity to human CB2 receptor and rat CB2 receptor with Ki of 422 nM and 238 nM. MDA7 exhibits analgesic activity in rats models.
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- No. CAS: 1103840-28-3
- Fòrmula: C22H25NO2
- Peso molecular:335.44
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Actividad biológica
Descripciòn
IC50 & Target
|
rat CB2-R 67.4 nM (IC50) |
hCB2-R 128 nM (IC50) |
rat CB2-R 238 nM (Ki) |
hCB2-R 422 nM (Ki) |
rCB1-R 2565 nM (Ki) |
Chemical Information
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No. CAS 1103840-28-3
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Peso molecular 335.44
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Fòrmula C22H25NO2
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SMILES
O=C(N1CCCCC1)C2=CC=C3C(OCC3(CC4=CC=CC=C4)C)=C2
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)