TYK2 - tyrosine kinase 2 Gene
Species: Felis catus
Gene Type: protein coding
Gene ID: 101090171
TYK2 Products (4)
| mRNA | Protein | Name |
|---|---|---|
| XM_045045399.1 | XP_044901334.1 | non-receptor tyrosine-protein kinase TYK2 isoform X1 |
| XM_045045398.1 | XP_044901333.1 | non-receptor tyrosine-protein kinase TYK2 isoform X1 |
| XM_045045401.1 | XP_044901336.1 | non-receptor tyrosine-protein kinase TYK2 isoform X2 |
| XM_045045400.1 | XP_044901335.1 | non-receptor tyrosine-protein kinase TYK2 isoform X1 |
| Protein Preferred Names | Protein Names | |
|---|---|---|
|
non-receptor tyrosine-protein kinase TYK2 |
|
Related Agents
- Approval
- Clinical Phase
- Pre-clinical Phase
Approval
Bioactive Molecules
(19)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-50856 | Ruxolitinib | Inhibitor | 99.99% | Yes |
| HY-19569 | Upadacitinib | Inhibitor | 99.98% | Yes |
| HY-15315 | Baricitinib | Inhibitor | 99.97% | Yes |
| HY-117287 | Deucravacitinib | Inhibitor | 99.93% | Unkown |
| HY-50858 | Ruxolitinib phosphate | Inhibitor | 99.92% | Yes |
| HY-16379 | Pacritinib | Inhibitor | 99.93% | Yes |
| HY-107429 | Abrocitinib | Inhibitor | 99.26% | Unkown |
| HY-18300 | Filgotinib | Inhibitor | 99.77% | Yes |
| HY-19568 | Peficitinib | Inhibitor | 99.43% | Yes |
| HY-15315A | Baricitinib phosphate | Inhibitor | 99.97% | Yes |
| HY-109053 | Delgocitinib | Inhibitor | 99.61% | Unkown |
| HY-13577 | Oclacitinib | Inhibitor | 99.03% | Unkown |
| HY-13577A | Oclacitinib monomaleate | Inhibitor | 99.87% | Unkown |
| HY-18300A | Filgotinib maleate | Inhibitor | 99.88% | Yes |
| HY-50859 | Ruxolitinib sulfate | Inhibitor | / | Unkown |
| HY-19569A | Upadacitinib tartrate tetrahydrate | Inhibitor | / | Unkown |
| HY-19568A | Peficitinib hydrobromide | Inhibitor | / | Unkown |
| HY-16379A | Pacritinib hydrochloride | Inhibitor | / | Unkown |
| HY-19568B | Peficitinib hydrochloride | Inhibitor | / | Unkown |
Clinical Phase
Bioactive Molecules
(12)
| Cat. No. | Product Name |
Effect
|
Purity |
Phase |
|---|---|---|---|---|
| HY-112724 | Ivarmacitinib | Inhibitor | 99.62% | Phase 4 |
| HY-15999 | Cerdulatinib | Inhibitor | 99.06% | Phase 3 |
| HY-12469 | Decernotinib | Inhibitor | 99.91% | Phase 3 |
| HY-174905 | Quecitinib | Inhibitor | 99.35% | Phase 3 |
| HY-13034 | Gandotinib | Inhibitor | 99.86% | Phase 2 |
| HY-15270 | BMS-911543 | Inhibitor | 98.23% | Phase 2 |
| HY-156961 | Cadefrecitinib | Inhibitor | 99.81% | Phase 2 |
| HY-160144S | Lomedeucitinib | Inhibitor | 99.75% | Phase 2 |
| HY-19631 | Ilginatinib maleate | Inhibitor | 99.33% | Phase 2 |
| HY-159536 | Frevecitinib | Inhibitor | 99.42% | Phase 2 |
| HY-131968 | BMS-986202 | Inhibitor | 99.29% | Phase 1 |
| HY-101024 | PF-06263276 | Inhibitor | ≥99.0% | Phase 1 |
Pre-clinical Phase
Bioactive Molecules
(66)
| Cat. No. | Product Name |
Effect
|
Purity |
Rare Diseases
|
|---|---|---|---|---|
| HY-14435 | Pyridone 6 | Inhibitor | 98.20% | Unkown |
| HY-14722 | NVP-BSK805 | Inhibitor | 99.30% | Unkown |
| HY-19631A | Ilginatinib | Inhibitor | 99.81% | Unkown |
| HY-100895 | SAR-20347 | Inhibitor | 97.27% | Unkown |
| HY-113787 | (R)-9b | Inhibitor | 99.51% | Unkown |
| HY-158142 | PROTAC TYK2 degrader-1 | Degrader | 99.55% | Unkown |
| HY-153701S | Envudeucitinibum | Inhibitor | 99.56% | Unkown |
| HY-173357 | TYD-68 | Degrader | 99.54% | Unkown |
| HY-16640 | TCJL37 | Inhibitor | 99.89% | Unkown |
| HY-14722A | NVP-BSK805 dihydrochloride | Inhibitor | 99.36% | Unkown |
| HY-126242S | Tyk2-IN-7 | Inhibitor | 99.58% | Unkown |
| HY-101762 | TyK2-IN-2 | Inhibitor | 99.05% | Unkown |
| HY-15999A | Cerdulatinib hydrochloride | Inhibitor | 98.96% | Yes |
| HY-111745 | Tyk2-IN-5 | Inhibitor | 99.35% | Unkown |
| HY-131906 | JAK2-IN-7 | Inhibitor | 98.31% | Unkown |
| HY-150720 | TYK2-IN-12 | Inhibitor | 98.81% | Unkown |
| HY-19631B | Ilginatinib hydrochloride | Inhibitor | 98.92% | Unkown |
| HY-120469 | 2,6-Dichloro-N-(2-(cyclopropanecarboxamido)pyridin-4-yl)benzamide | Inhibitor | 99.80% | Unkown |
| HY-153440 | Methyl 6-(1-(4-methoxybenzyl)-1H-pyrazol-4-yl)-4-oxo-4,5-dihydropyrazolo[1,5-a]pyrazine-2-carboxylate | Inhibitor | 98.01% | Unkown |
| HY-111750 | JAK-IN-3 | Inhibitor | 98.92% | Unkown |
| HY-126141 | JAK/HDAC-IN-1 | Inhibitor | 98.63% | Unkown |
| HY-13961 | GLPG0634 analog | Inhibitor | 98.07% | Unkown |
| HY-152080 | Blovacitinib | Inhibitor | 99.71% | Unkown |
| HY-170772 | Dual Cathepsin L/JAK-IN-1 | Inhibitor | 98.47% | Unkown |
| HY-143884 | JAK2/TYK2-IN-1 | Inhibitor | 99.94% | Unkown |
| HY-148060 | JAK-IN-21 | Inhibitor | 99.72% | Unkown |
| HY-18710 | BMS-066 | Inhibitor | 99.09% | Unkown |
| HY-18315 | Bayer-18 | Inhibitor | / | Unkown |
| HY-14722C | NVP-BSK805 trihydrochloride | Inhibitor | / | Unkown |
| HY-184075S | Nomelcitinib | Inhibitor | / | Unkown |
| HY-187211 | TYK2 activator-2 | Modulator | / | Unkown |
| HY-174430 | WWQ-131 | Inhibitor | / | Unkown |
| HY-147754 | JAK3/BTK-IN-6 | Inhibitor | / | Unkown |
| HY-N14094 | Tubulosine | Inhibitor | / | Unkown |
| HY-178282 | JAK1-IN-19 | Inhibitor | / | Unkown |
| HY-153058 | LRRK2-IN-8 | Inhibitor | / | Unkown |
| HY-149283 | JAK/HDAC-IN-2 | Inhibitor | / | Unkown |
| HY-175983 | JAK1/TYK2-IN-5 | Inhibitor | / | Unkown |
| HY-143885 | JAK1/TYK2-IN-3 | Inhibitor | / | Unkown |
| HY-163304 | Tyk2-IN-16 | Inhibitor | / | Unkown |
| HY-177131 | Soficitinib | Inhibitor | 98.54% | Unkown |
| HY-153103 | LRRK2/NUAK1/TYK2-IN-1 | Inhibitor | / | Unkown |
| HY-177130S | Socrodeucitinib | Inhibitor | / | Unkown |
| HY-154994 | JAK-IN-30 | Inhibitor | / | Unkown |
| HY-18709 | Tyk2-IN-3 | Inhibitor | / | Unkown |
| HY-175310S | Voderdeucitinib | Inhibitor | / | Unkown |
| HY-181278 | Deucravacitinib analog 1 | / | Unkown | |
| HY-149296 | JAK1-IN-12 | Inhibitor | / | Unkown |
| HY-175684 | JAK2-IN-14 | Inhibitor | / | Unkown |
| HY-168269 | Tyk2-IN-20 | Inhibitor | / | Unkown |
| HY-176793 | Embricitinib | Inhibitor | / | Unkown |
| HY-401428 | TYK2 ligand 3 | Degrader | / | Unkown |
| HY-173359 | TYK2 ligand 2 | Ligand | / | Unkown |
| HY-158692 | Tyk2-IN-18 | Inhibitor | / | Unkown |
| HY-168339 | Tyk2-IN-22 | Inhibitor | / | Unkown |
| HY-188034 | JAK-IN-44 | Inhibitor | / | Unkown |
| HY-112783 | TYK2 ligand 4 | Ligand | / | Unkown |
| HY-158340 | TYK2 ligand 1 | Inhibitor | / | Unkown |
| HY-162862 | JAK-IN-38 | Inducer | / | Unkown |
| HY-184786 | Tyk2-IN-14 | Inhibitor | / | Unkown |
| HY-123187 | AS2553627 | Inhibitor | / | Unkown |
| HY-184866 | Tyk2-IN-26 | Inhibitor | / | Unkown |
| HY-157121 | JAK-IN-34 | Inhibitor | / | Unkown |
| HY-162862 | JAK-IN-38 | Inhibitor | / | Unkown |
| HY-123939 | JAK1/3-IN-1 | Inhibitor | / | Unkown |
| HY-184833 | Tyk2-IN-25 | Inhibitor | / | Unkown |