GPCR agonist-2
Based on 1 Customer Validation
GPCR agonist-2 (Compound 5j) is a GPCR GPR109b (HM74) agonist, with a pEC50 value of 6.51. GPCR agonist-2 can be used for research of lipid disorders.
For research use only. We do not sell to patients.
- Purity: 99.93%
- CAS No.: 291528-35-3
- Formula: C10H10N2O4
- Molecular Weight:222.20
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Storage:
4°C, protect from light
* In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
Biological Activity
Chemical Information
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CAS No. 291528-35-3
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Appearance Solid
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Molecular Weight 222.20
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Formula C10H10N2O4
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Color Light yellow to yellow
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SMILES
O=C(O)C1=CC=C(NC2CC2)C([N+]([O-])=O)=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
4°C, protect from light
* In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
Solvent & Solubility
DMSO : 125 mg/mL (562.56 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (270 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 4.5005 mL | 22.5023 mL | 45.0045 mL | 112.5113 mL |
| 5 mM | 0.9001 mL | 4.5005 mL | 9.0009 mL | 22.5023 mL | |
| 10 mM | 0.4500 mL | 2.2502 mL | 4.5005 mL | 11.2511 mL | |
| 15 mM | 0.3000 mL | 1.5002 mL | 3.0003 mL | 7.5008 mL | |
| 20 mM | 0.2250 mL | 1.1251 mL | 2.2502 mL | 5.6256 mL | |
| 25 mM | 0.1800 mL | 0.9001 mL | 1.8002 mL | 4.5005 mL | |
| 30 mM | 0.1500 mL | 0.7501 mL | 1.5002 mL | 3.7504 mL | |
| 40 mM | 0.1125 mL | 0.5626 mL | 1.1251 mL | 2.8128 mL | |
| 50 mM | 0.0900 mL | 0.4500 mL | 0.9001 mL | 2.2502 mL | |
| 60 mM | 0.0750 mL | 0.3750 mL | 0.7501 mL | 1.8752 mL | |
| 80 mM | 0.0563 mL | 0.2813 mL | 0.5626 mL | 1.4064 mL | |
| 100 mM | 0.0450 mL | 0.2250 mL | 0.4500 mL | 1.1251 mL |