GPR17 agonist 2
GPR17 agonist 2 (compound 10) is a human GPR17 agonist and selective P2Y receptor non-activator.GPR17 agonist 2 modulates intracellular cAMP levels through functional activation of its target receptor.GPR17 agonist 2 can be used for the research of multiple sclerosis, cerebral ischemia, traumatic brain injury, spinal cord injury.
For research use only. We do not sell to patients.
- Formula: C19H32Cl2N9O12P3
- Molecular Weight:742.34
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
GPR17 agonist 2 (compound 10) (dose-response curve for EC50 determination) is a potent, full agonist of human GPR17 in HEK293 L9-2 cells, with an EC50 of 62 pM, and shows high selectivity for human GPR17 over human P2Y12, P2Y13, and P2Y14 receptors[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Molecular Weight 742.34
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Formula C19H32Cl2N9O12P3
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SMILES
O=P(OP(C(Cl)(Cl)P([O-])([O-])=O)([O-])=O)([O-])OC[C@@H]1[C@@H](O)[C@@H](O)[C@H](N2C=NC3=C(N)N=C(C#CC4=CC=CC=C4)N=C32)O1.[NH4+].[NH4+].[NH4+].[NH4+]
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
GPR17 agonist 2 Related Classifications
HY-181738 Related Classifications
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