GSK-2250665A
Based on 1 Customer Validation
GSK-2250665A (Compound 13) is a selective Itk inhibitor with a pKi of 9.2.
For research use only. We do not sell to patients.
- Purity: 96.35%
- CAS No.: 1246030-96-5
- Formula: C26H29N5OS
- Molecular Weight:459.61
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Storage:
Store at room temperature, keep dry and cool.
In solvent -80°C, 1 year , -20°C, 6 months
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
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Immunology/Inflammation Compound Library
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Kinase Inhibitor Library
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Protein Tyrosine Kinase Compound Library
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Highly Selective Inhibitors Library
HY-L158
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Serine/Threonine Kinase Inhibitor Library
HY-L164
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Bioactive Compound Library Max
HY-L181
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MCE Bioactive Compound Library
HY-L001V
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Bioactive Compound Library
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Protein Kinase Compound Library
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High-Throughput Bioactive Compound Library
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Biological Activity
GSK-2250665A (Compound 13) achieves a pIC50 of 7.3 in the cell assay, measuring inhibition of IFNγ production from PBMCs (Peripheral Blood Mononuclear Cells) [1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 1246030-96-5
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Appearance Solid
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Molecular Weight 459.61
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Formula C26H29N5OS
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Color White to off-white
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SMILES
CCC1=CC=C2C(SC(NC3=NC(N[C@H]4CC[C@@H](CC4)O)=NC(CC5=CC=CC=C5)=C3)=N2)=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Store at room temperature, keep dry and cool
In solvent -80°C 1 year -20°C 6 months
Purity & Documentation
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Data Sheet (268 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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Handling Instructions (2659 KB)
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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