2. Membrane Transporter/Ion Channel
  3. HCN Channel
  4. HCN2-IN-4

HCN2-IN-4 is an orally active HCN2 ion channel inhibitor, with an IC50 of 3 nM. HCN2-IN-4 inhibits the activity of HCN2 ion channels. HCN2-IN-4 can be used in the research of pain, tinnitus and central nervous system diseases.

For research use only. We do not sell to patients.

HCN2-IN-4

HCN2-IN-4 Chemical Structure

CAS No. : 3080809-13-5

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Other Forms of HCN2-IN-4:

HCN2-IN-4 Related Antibodies

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Description

HCN2-IN-4 is an orally active HCN2 ion channel inhibitor, with an IC50 of 3 nM. HCN2-IN-4 inhibits the activity of HCN2 ion channels. HCN2-IN-4 can be used in the research of pain, tinnitus and central nervous system diseases[1].

In Vitro

HCN2-IN-4 (Compound 49) potently and selectively inhibits human HCN2 channels, with an IC50 of 3 nM[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

HCN2-IN-4 Related Antibodies
Molecular Weight

455.46

Formula

C21H18FN5O4S
CAS No.
SMILES

O=C(C1=CC=NS1)NC2=NN(C[C@@H](C)OC)C3=NC=C(C4=CC=C(OCO5)C5=C4F)C=C23
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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HCN2-IN-4 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

HCN2-IN-43080809-13-5HCN ChannelHyperpolarization activated cyclic nucleotide gated channelsHCN2 ion channel inhibitorpaintinnitus and central nervous system diseasesInhibitorinhibitorinhibit

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