HCN2-IN-4
HCN2-IN-4 is an orally active HCN2 ion channel inhibitor, with an IC50 of 3 nM. HCN2-IN-4 inhibits the activity of HCN2 ion channels. HCN2-IN-4 can be used in the research of pain, tinnitus and central nervous system diseases.
For research use only. We do not sell to patients.
- CAS No.: 3080809-13-5
- Formula: C21H18FN5O4S
- Molecular Weight:455.46
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
HCN2-IN-4 (Compound 49) potently and selectively inhibits human HCN2 channels, with an IC50 of 3 nM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3080809-13-5
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Molecular Weight 455.46
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Formula C21H18FN5O4S
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SMILES
O=C(C1=CC=NS1)NC2=NN(C[C@@H](C)OC)C3=NC=C(C4=CC=C(OCO5)C5=C4F)C=C23
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)