HIPK4-IN-1
HIPK4-IN-1 is a HIPK4 inhibitor (IC50 = 0.12 μM). HIPK4-IN-1 causes almost no HIPK4 degradation. HIPK4-IN-1 can be used for research on sperm development.
For research use only. We do not sell to patients.
- Formula: C20H19N3O4
- Molecular Weight:365.38
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
IC50 & Target
[1]|
HIPK4 0.12 μM (IC50) |
Cellular Effect
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HEK-293T | IC50 |
2.9 μM
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Target engagement against NanoLuc-HIPK4 in HEK293T cells assessed by NanoBRET competitive displacement of a cell-permeable tracer.
Target engagement against NanoLuc-HIPK4 in HEK293T cells assessed by NanoBRET competitive displacement of a cell-permeable tracer.
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42182270 |
In Vitro
HIPK4-IN-1 engages NanoLuc-HIPK4 in HEK293T cells with a NanoBRET IC50 of 2.9 μM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Molecular Weight 365.38
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Formula C20H19N3O4
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SMILES
COC1=C(OC)C=C2C(NC3=C(OC)C=CC=C3OC)=C(C#N)C=NC2=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
HIPK4-IN-1 Related Classifications
HY-190749 Related Classifications
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