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Cat. No.: HY-101718R

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Aticaprant (Standard)

(Synonyms: CERC-501 (Standard); LY-2456302 (Standard))

Aticaprant (Standard) (CERC-501 (Standard)) is the analytical standard of Aticaprant (HY-101718). This product is intended for research and analytical applications. Aticaprant (CERC-501) is a potent and centrally-penetrant kappa opioid receptor antagonist with a K_i of 0.807 nM.

For research use only. We do not sell to patients.

CAS No.: 1174130-61-0
Formula: C₂₆H₂₇FN₂O₂
Molecular Weight:418.50

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Aticaprant (Standard) Chemical Structure

CAS No.: 1174130-61-0

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

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- Application
Chemical Information
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Bioz

Product Information

Information

Application

The compound is the grade of analytical standard, which is the reference standard supplied assay. It is commonly used in qualitative, quantitative and methodological research experiments in HPLC, GC and MS.

Chemical Information

CAS No. 1174130-61-0
Molecular Weight 418.50
Formula C₂₆H₂₇FN₂O₂
SMILES

O=C(N)C1=CC=C(OC2=CC=C(CN3[C@H](C4=CC(C)=CC(C)=C4)CCC3)C=C2)C(F)=C1
Synonyms

CERC-501 (Standard); LY-2456302 (Standard)
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

References

[1]. Rorick-Kehn LM, et al. LY2456302 is a novel, potent, orally-bioavailable small molecule kappa-selective antagonist with activity in animal models predictive of efficacy in mood and addictive disorders. Neuropharmacology. 2014 Feb;77:131-44. [Content Brief]

[2]. Jackson KJ, et al. Effects of orally-bioavailable short-acting kappa opioid receptor-selective antagonist LY2456302on nicotine withdrawal in mice. Neuropharmacology. 2015 Oct;97:270-4. [Content Brief]

Calculators

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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