1. Metabolic Enzyme/Protease
  2. Glucokinase
  3. IHVR-11029

IHVR-11029 is a small molecule inhibitor of ER α-glucosidases, with an EC50 of 0.09 μM.

For research use only. We do not sell to patients.

IHVR-11029 Chemical Structure

IHVR-11029 Chemical Structure

CAS No. : 1383152-30-4

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5 mg USD 160 In-stock
10 mg USD 250 In-stock
25 mg USD 550 In-stock
50 mg USD 950 In-stock
100 mg USD 1550 In-stock
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Based on 1 publication(s) in Google Scholar

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Description

IHVR-11029 is a small molecule inhibitor of ER α-glucosidases, with an EC50 of 0.09 μM[1].

IC50 & Target

EC50: 0.09 μM (ER α-glucosidases)[1].

In Vitro

IHVR-11029 exhibits EC50 values of 1.3 μM, 3.3 μM and 0.75 μM for BVDV, TARV and DENV, respectively.

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

375.41

Formula

C18H27F2NO5

CAS No.
Appearance

Solid

Color

White to off-white

SMILES

OC[C@@H]1[C@@H](O)[C@H](O)[C@@H](O)CN1CCCCCCOC2=CC(F)=CC=C2F

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, protect from light, stored under nitrogen

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light, stored under nitrogen)

Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (266.38 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.6638 mL 13.3188 mL 26.6375 mL
5 mM 0.5328 mL 2.6638 mL 5.3275 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light, stored under nitrogen). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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In Vivo Dissolution Calculator
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Calculation results:
Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light, stored under nitrogen). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.6638 mL 13.3188 mL 26.6375 mL 66.5939 mL
5 mM 0.5328 mL 2.6638 mL 5.3275 mL 13.3188 mL
10 mM 0.2664 mL 1.3319 mL 2.6638 mL 6.6594 mL
15 mM 0.1776 mL 0.8879 mL 1.7758 mL 4.4396 mL
20 mM 0.1332 mL 0.6659 mL 1.3319 mL 3.3297 mL
25 mM 0.1066 mL 0.5328 mL 1.0655 mL 2.6638 mL
30 mM 0.0888 mL 0.4440 mL 0.8879 mL 2.2198 mL
40 mM 0.0666 mL 0.3330 mL 0.6659 mL 1.6648 mL
50 mM 0.0533 mL 0.2664 mL 0.5328 mL 1.3319 mL
60 mM 0.0444 mL 0.2220 mL 0.4440 mL 1.1099 mL
80 mM 0.0333 mL 0.1665 mL 0.3330 mL 0.8324 mL
100 mM 0.0266 mL 0.1332 mL 0.2664 mL 0.6659 mL
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IHVR-11029 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
IHVR-11029
Cat. No.:
HY-117721
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