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TM471-1

TM471-1 is an orally active and covalent Bruton's tyrosine kinase (BTK) inhibitor with IC50 values of 1.3 nM (BTKWT), >40,000 nM (BTKC481S), 7.9 nM (TEC) and 12.4 nM (TXK). TM471-1 inhibits cell growth in vivo and in vitro, arrests cell cycle at G0/G1 phase and induces cell apoptosis.

For research use only. We do not sell to patients.

  • CAS No.: 2649008-95-5
  • Formula: C27H29N5O3
  • Molecular Weight:471.55
  • Storage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

  • TM471-1 Chemical Structure
    TM471-1 Chemical Structure
CAS No.: 2649008-95-5
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609-228-6898
[email protected] [email protected]
Find Your Local Distributor Your local distributor: Hycultec GmbHHycultec
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  • TM471-1 Chemical Structure
    TM471-1 Chemical Structure
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  • TM471-1