Deschlorodiazepam
Based on 1 Customer Validation
Deschlorodiazepam is an analytical reference standard categorized as a benzodiazepine.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度: 98.64%
- CAS 番号: 3034-65-9
- 分子式: C16H14N2O
- 分子量:250.30
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保管条件:
Store at room temperature 3 years.
In solvent -80°C, 2 years , -20°C, 1 year
生物活性
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| Sf9 | IC50 |
>10 μM
Compound: figure 3, R4C1
|
Displacement of [3H]Ro15-4513 from GABAA alpha-1-beta-2-gamma-2 receptor expressed in Sf9 baculovirus system
Displacement of [3H]Ro15-4513 from GABAA alpha-1-beta-2-gamma-2 receptor expressed in Sf9 baculovirus system
|
[PMID: 18537233] |
| Sf9 | IC50 |
>10 μM
Compound: figure 3, R4C1
|
Displacement of [3H]Ro15-4513 from GABAA alpha-5-beta-2-gamma-2 receptor expressed in Sf9 baculovirus system
Displacement of [3H]Ro15-4513 from GABAA alpha-5-beta-2-gamma-2 receptor expressed in Sf9 baculovirus system
|
[PMID: 18537233] |
化学情報
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CAS 番号 3034-65-9
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性状 Solid
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分子量 250.30
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分子式 C16H14N2O
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Color Light yellow to brown
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SMILES
O=C1N(C)C2=C(C(C3=CC=CC=C3)=NC1)C=CC=C2
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Store at room temperature 3 years
In solvent -80°C 2 years -20°C 1 year
溶剤 & 溶解度
DMSO : 25 mg/mL (99.88 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 2 years; -20°C, 1 year. When stored at -80°C, please use it within 2 years. When stored at -20°C, please use it within 1 year.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 2 years; -20°C, 1 year. When stored at -80°C, please use it within 2 years. When stored at -20°C, please use it within 1 year.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (275 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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取扱説明書 (2659 KB)
参考文献
[1]. Basile AS, et al. Brain concentrations of benzodiazepines are elevated in an animal model of hepatic encephalopathy. Proc Natl Acad Sci U S A. 1990 Jul;87(14):5263-7. [Content Brief]
[2]. Sternbach LH, et al. Quinazolines and 1,4-benzodiazepines. 64. Comparison of the stereochemistry of diazepam with that of close analogs with marginal biological activity. J Med Chem. 1974 Mar;17(3):374-7. [Content Brief]
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 2 years; -20°C, 1 year. When stored at -80°C, please use it within 2 years. When stored at -20°C, please use it within 1 year.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 3.9952 mL | 19.9760 mL | 39.9521 mL | 99.8801 mL |
| 5 mM | 0.7990 mL | 3.9952 mL | 7.9904 mL | 19.9760 mL | |
| 10 mM | 0.3995 mL | 1.9976 mL | 3.9952 mL | 9.9880 mL | |
| 15 mM | 0.2663 mL | 1.3317 mL | 2.6635 mL | 6.6587 mL | |
| 20 mM | 0.1998 mL | 0.9988 mL | 1.9976 mL | 4.9940 mL | |
| 25 mM | 0.1598 mL | 0.7990 mL | 1.5981 mL | 3.9952 mL | |
| 30 mM | 0.1332 mL | 0.6659 mL | 1.3317 mL | 3.3293 mL | |
| 40 mM | 0.0999 mL | 0.4994 mL | 0.9988 mL | 2.4970 mL | |
| 50 mM | 0.0799 mL | 0.3995 mL | 0.7990 mL | 1.9976 mL | |
| 60 mM | 0.0666 mL | 0.3329 mL | 0.6659 mL | 1.6647 mL | |
| 80 mM | 0.0499 mL | 0.2497 mL | 0.4994 mL | 1.2485 mL |