DPP-4-IN-3
DPP-4-IN-3 (Compound 5a) is a potent dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 of 0.75 nM. DPP-4-IN-3 shows excellent antioxidant and insulinotropic activity.
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研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 2402735-14-0
- 分子式: C19H22N6O2
- 分子量:366.42
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
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DPP-4 |
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| INS1(832/13) | IC50 |
0.0028 μM
Compound: 5a
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Antidiabetic activity in glucose-treated rat INS1(832/13) cells assessed as increase in insulin release in presence of 3 mM glucose measured after 2 hrs by radioimmunoassay
Antidiabetic activity in glucose-treated rat INS1(832/13) cells assessed as increase in insulin release in presence of 3 mM glucose measured after 2 hrs by radioimmunoassay
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[PMID: 31812034] |
化学情報
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CAS 番号 2402735-14-0
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分子量 366.42
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分子式 C19H22N6O2
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SMILES
CCOC(N1CCN(CC1)C2=NN3C(C=C2)=NN=C3C4=CC=CC(C)=C4)=O
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
DPP-4-IN-3 関連分類
HY-146455 関連分類
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