FGH31
FGH31 (Compound 24) is a potent, selective, GRK2 dependency dopamine D4 agonist, with the Ki of 1.6 nM. FGH31 partial activates β- arrestin.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 3033813-47-4
- 分子式: C33H36N4O2
- 分子量:520.66
-
保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
生物活性
-
化学情報
- 純度とドキュメンテーション
- 参考文献
-
Help & FAQs
生物活性
|
Dopamine D4 receptor 1.6 nM (Ki) |
GRK2 |
FGH31 (Compound 24) (50 μM) decreases at a similar rate as Imipramine (HY-B1490A) in rat liver microsomes[1].
FGH31 (50 μM, 4 h) shows no significant transport by P-glycoprotein (P-gp) in Caco-2 cells[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
-
CAS 番号 3033813-47-4
-
分子量 520.66
-
分子式 C33H36N4O2
-
SMILES
O=C(NCCCN1CCN(C2=CC=CC=C2OC)CC1)NC3=CC=CC=C3C4=CC=C(C5=CC=CC=C5)C=C4
-
輸送条件
Room temperature in continental US; may vary elsewhere.
-
保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
FGH31 関連分類
HY-155099 関連分類
Powered by Bioz