Ocaperidone (Standard)
Ocaperidone (Standard) is the analytical standard of Ocaperidone (HY-101094). This product is intended for research and analytical applications. Ocaperidone is an effective antipsychotic agent, acting as a potent 5-HT2 and dopamine D2 antagonist, and a 5-HT1A agonist, with Kis of 0.14 nM, 0.46 nM, 0.75 nM, 1.6 nM and 5.4 nM for 5-HT2, a1-adrenergic receptor, dopamine D2, histamine H1 and a2-adrenergic receptor, respectively, and a pEC50 and pKi of 7.60 and 8.08 for h5-HT1A.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 129029-23-8
- 分子式: C24H25FN4O2
- 分子量:420.48
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Product Information
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化学情報
- 純度とドキュメンテーション
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Help & FAQs
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HY-101094
Ocaperidone5-HT2/Dopamine D2 Antagonist -
HY-B0032A
Lurasidone -
HY-14542
Ziprasidone5-HT/DA Receptor Antagonist -
HY-15414
VortioxetineSerotonin Transporter Inhibitor -
HY-B0031
Quetiapine hemifumarate5-HT Agonist/D2 Antagonist -
HY-N0145
Puerarin5-HT Receptor Antagonist -
HY-112061
8-OH-DPAT5-HT Receptor Agonist -
HY-14544
Quetiapine5-HT Agonist/D2 Antagonist -
HY-14262
VilazodoneSerotonin Reuptake Inhibitor -
HY-B0031R
Quetiapine hemifumarate (Standard) -
HY-103093
ZotepineAntipsychotic Agent -
HY-N0145R
Puerarin (Standard)5-HT Receptor Antagonist
Product Information
説明
アプリケーション
The compound is the grade of analytical standard, which is the reference standard supplied assay. It is commonly used in qualitative, quantitative and methodological research experiments in HPLC, GC and MS.
化学情報
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CAS 番号 129029-23-8
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分子量 420.48
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分子式 C24H25FN4O2
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SMILES
O=C1C(CCN2CCC(C3=NOC4=C3C=CC(F)=C4)CC2)=C(C)N=C5N1C=CC=C5C
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別名
R79598 (Standard)
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
[1]. Leysen JE, et al. In vitro and in vivo receptor binding and effects on monoamine turnover in rat brain regions of the novel antipsychotics risperidone and ocaperidone. Mol Pharmacol. 1992 Mar;41(3):494-508. [Content Brief]
[2]. Cosi C, et al. Agonist, antagonist, and inverse agonist properties of antipsychotics at human recombinant 5-HT(1A) receptors expressed in HeLa cells. Eur J Pharmacol. 2001 Dec 14;433(1):55-62. [Content Brief]
[3]. Rijnders HJ, et al. The discriminative stimulus properties of buspirone involve dopamine-2 receptor antagonist activity. Psychopharmacology (Berl). 1993;111(1):55-61. [Content Brief]
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
Ocaperidone (Standard) 関連分類
HY-101094R 関連分類
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