PD-149164
PD-149164 is a potent agonist of cholecystokinin B (CCK-B) receptor, with IC50 values of 0.083 nM and 75 nM in binding assay to CCK-B and CCK-A.
For research use only. We do not sell to patients.
- CAS No.: 181941-32-2
- Formula: C33H38FN3O5
- Molecular Weight:575.67
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Protocols
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
IC50 & Target
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CCKAR 75 nM (IC50) |
CCKBR 0.083 nM (IC50) |
Chemical Information
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CAS No. 181941-32-2
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Molecular Weight 575.67
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Formula C33H38FN3O5
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SMILES
O=C(C[C@H](CC1=CC=C(C=C1)F)NC([C@@](NC(OC2C3CC4CC(CC2C4)C3)=O)(C)CC5=CNC6=C5C=CC=C6)=O)O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Protocols
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Cell Cytotoxicity Assay
Cytotoxicity assays are usually based on the assessment of cell membrane damage, which can also be indirectly detected by measuring cell viability. Detection methods include MTT assay, CKK-8 assay, LDH assay and ATP assay, etc.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
PD-149164 Related Classifications
HY-123434 Related Classifications
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