(±)-Befunolol
Based on 1 publication(s) in Google Scholar
(±)-Befunolol is a β-adrenoceptor blocking agent.
연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.
- CAS No.: 39552-01-7
- 화학식: C16H21NO4
- 분자량:291.34
-
보관:
Please store the product under the recommended conditions in the Certificate of Analysis.
Publications Citing Use of MedChemExpress (MCE) (±)-Befunolol
MoreAll Adrenergic Receptor Isoforms
More
Biological Activity
제품 설명
IC50 & Target
Adrenoreceptor[1]
In Vitro
A β-adrenoceptor blocking agent, Befunolol, is found to has intrinsic sympathomimetic activities in isolated right atria, trachea and taenia caecum of guinea pig (intrinsic activities are 0.22-0.28). The pD2-values of Befunolol estimated in the isolated organs are significantly different from its pA2-values against isoprenaline. Befunolol interacts with the beta-adrenoceptor where there may be two different sites: one site for agonistic action and the other for competitive antagonistic action. The intrinsic activity of Befunolol may be equal to its selectivity for both the sites[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. .
Chemical Information
-
CAS No. 39552-01-7
-
분자량 291.34
-
화학식 C16H21NO4
-
SMILES
CC(C1=CC2=CC=CC(OCC(O)CNC(C)C)=C2O1)=O
-
선적
Room temperature in continental US; may vary elsewhere.
-
보관
Please store the product under the recommended conditions in the Certificate of Analysis.
Publications (1)
-
Journal Impact Factor
-
Most Recent
-
J Pharm Biomed Anal
Screening method of mildronate and over 300 doping agents by reversed-phase liquid chromatography-high resolution mass spectrometry. [Abstract]2021 Feb 20:195:113870. PMID: 33453569
순도&문서
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)