FGH31
FGH31 (Compound 24) is a potent, selective, GRK2 dependency dopamine D4 agonist, with the Ki of 1.6 nM. FGH31 partial activates β- arrestin.
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- CAS No.: 3033813-47-4
- 화학식: C33H36N4O2
- 분자량:520.66
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보관:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- 순도&문서
- References
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Help & FAQs
Biological Activity
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Dopamine D4 receptor 1.6 nM (Ki) |
GRK2 |
FGH31 (Compound 24) (50 μM) decreases at a similar rate as Imipramine (HY-B1490A) in rat liver microsomes[1].
FGH31 (50 μM, 4 h) shows no significant transport by P-glycoprotein (P-gp) in Caco-2 cells[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3033813-47-4
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분자량 520.66
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화학식 C33H36N4O2
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SMILES
O=C(NCCCN1CCN(C2=CC=CC=C2OC)CC1)NC3=CC=CC=C3C4=CC=C(C5=CC=CC=C5)C=C4
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
FGH31 Related Classifications
HY-155099 Related Classifications
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