PD-161182
PD-161182 is a non-peptide NK-3 antagonist. PD-161182 can be studied in NK-3-related central nervous system disturbances, pain, inflammation, pulmonary and skin diseases.
연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.
- CAS No.: 168570-35-2
- 화학식: C29H40F2N4O4
- 분자량:546.65
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보관:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
제품 설명
Cellular Effect
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| CHO | IC50 |
1400 nM
Compound: 61
|
Compound was tested for the inhibition of [125I]-[MePhe7]-NKB binding to cloned human Tachykinin receptor 3 in CHO cell lines
Compound was tested for the inhibition of [125I]-[MePhe7]-NKB binding to cloned human Tachykinin receptor 3 in CHO cell lines
|
[PMID: 8648606] |
Chemical Information
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CAS No. 168570-35-2
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분자량 546.65
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화학식 C29H40F2N4O4
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SMILES
O=C(N[C@](C)(C(NCCCCCCCNC(N)=O)=O)CC1=CC=CC(F)=C1F)O[C@@H](C(C)C)C2=CC=CC=C2
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)