country

Change Language

EN - English
FR - Français
DE - Deutsch
ES - Español
JA - 日本語
KO - 한국어

Country or Region:

United States

Product Name	Size / Unit Price	Qty

Total: USD 0.00 Checkout

Cat. No.: HY-P10878

Copy Link Print Information

UK140

UK140 is the inhibitor for urokinase-type plasminogen activator (uPA) with K_i of 0.20 µM and 2.79 µM for huPA anf muPA. UK140 can be used in metastasis-related research.

연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.

화학식: C₇₂H₁₀₅N₁₉O₂₅S₃
분자량:1732.91

보관:

Please store the product under the recommended conditions in the Certificate of Analysis.

UK140 Chemical Structure

Amount: USD 0.00

* 장바구니에 담기 전 물품의 수량을 선택해 주십시오.

Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- 제품 설명
- IC₅₀ & Target
Chemical Information
순도&문서
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

제품 설명

UK140 is the inhibitor for urokinase-type plasminogen activator (uPA) with K_i of 0.20 µM and 2.79 µM for huPA anf muPA. UK140 can be used in metastasis-related research^[1].

IC₅₀ & Target

K_i: 0.20 µM (huPA); 2.79 µM (muPA)

Chemical Information

분자량 1732.91

화학식 C₇₂H₁₀₅N₁₉O₂₅S₃

Sequence

Ala-Cys-Asn-Ser-Lys-Phe-Ser-Gly-Cys-Gly-Val-Asp-Pro-Ser-Ser-Cys-Gly (cyclized via TBMB and Cys2,9,16)

Sequence Shortening

ACNSKFSGCGVDPSSCG (cyclized via TBMB and Cys2,9,16)

선적

Room temperature in continental US; may vary elsewhere.

보관

Please store the product under the recommended conditions in the Certificate of Analysis.

순도&문서

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (258 KB)

COA (2659 KB)

Elemental Analysis Report (2659 KB)

HNMR (2659 KB)

CNMR (2659 KB)

RP-HPLC (2659 KB)

NP-HPLC (2659 KB)

MS (2659 KB)

LCMS (2659 KB)

IR (2659 KB)

GC (2659 KB)

OR (2659 KB)

SDS-PAGE (2659 KB)

SEC-HPLC (2659 KB)

Other Report (2659 KB)

Handling Instructions (2659 KB)

References

[1]. Mazzocato Y, et al., A novel genetically-encoded bicyclic peptide inhibitor of human urokinase-type plasminogen activator with better cross-reactivity toward the murine orthologue. Bioorg Med Chem. 2023 Nov 15;95:117499. [Content Brief]

Calculators

몰농도 계산기

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

=
Concentration Concentration

×
Volume Volume

×
Molecular Weight Molecular Weight

농도 희석 계산기

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

×

Volume _(start) Volume _(start)

=

Concentration _(final) Concentration _(final)

×

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

UK140 Related Classifications

HY-P10878 Related Classifications

Metabolic Enzyme/Protease

PAI-1

Disease Areas

Cancer

Peptides

Peptide and Derivatives

Inhibitors and Substrates

Cancer

Cancer Targeted Therapy Cancer Metabolism and Metastasis

Bioz

Powered by Bioz See more details on Bioz

Keywords

UK140
UK 140
UK-140
PAI-1
Inhibitor
inhibitor
inhibit

Your Recently Viewed Products

UK140

100 mg 견적 받기

Subscribe to the

MedChemExpress

Newsletter

Subscribe

MOQ

Minimum order quantity

100 mg

견적 받기 해외재고보유

Other size

견적 받기

Please select quantity

Amount: USD 0.00

Biological Activity

제품 설명

IC₅₀ & Target

Chemical Information

순도&문서

References

Sign in to MedChemExpress 로그인

Register

Sign in to MedChemExpress

Keep me logged in. 비밀번호 찾기

회원가입

At least 6 characters

Personalize your experience, you are currently not signed in. For a better experience, please create an online profile, you can:

Obtain points redemption prizes

Check out faster

Add multiple shipping locations

View orders

Assay Types

1/16

온라인 문의

Your information is safe with us. *Required Fields.

상품명 *
Field is required.

Requested Quantity *
Field is required.

고객명 *
Field is required.

호칭 *
Field is required.

이메일 *
Field is required.

Please enter a valid Email Address.

전화번호 *
Field is required.

Department

회사명 *
Field is required.

시
시

시

Enter Others City *
Field is required.

Field is required.

도 도 *
Field is required.

국가 또는 지역 *
Field is required.

Container *
Field is required.

MCE Japan Authorized Agent:

ナミキ商事株式会社コスモ・バイオ株式会社重松貿易株式会社

비고

Request for Report

Please fill out this form to request the report. We will send it to your Email address shortly.
Your information is safe with us. *Required Fields.

상품명 *
Field is required.

Lot # *
Field is required.

고객명 *
Field is required.

이메일 *
Field is required.

Please enter a valid Email Address.

전화번호
Field is required.

Department *
Field is required.

회사명 *
Field is required.

국가 또는 지역 *
Field is required.

비고

대량구매 문의 Request for Report 온라인 문의 고객리뷰 Request for Recombinant Proteins Catalog

We have received your request and will respond to you as soon as possible. Congratulations! Uh-oh!

We have received your inquiry regarding and will respond to you as soon as possible. We have received your request and will respond to you as soon as possible. Thank You for Your Feedback! This product is a controlled substance and not for sale in your territory. It appears that we were unable to send an email to . Please verify your email address and try again!

Inquiry Information

상품명:

Cat. No.:

수량:

MCE Japan Authorized Agent:

Inquiry Information

상품명:

CAS No.:

Species:

Purity:

수량:

Licensing Opportunities

Your information is safe with us. *Required Fields.

고객명 *
Field is required.

호칭 *
Field is required.

Role/Position *
Field is required.

회사명 *
Field is required.

국가 또는 지역 *
Field is required.

도 도 *
Field is required.

이메일 *
Field is required.

Please enter a valid Email Address.

전화번호 *
Field is required.

상품명
Field is required.

CAS No.
Field is required.

비고

MedChemExpress

MedChemExpress

Contact Us

About Us

Headquarters

Distributors

Statement on False Report

Careers

고객지원

고객지원

Technical Support

서비스

Ordering Information

편리한 반품

배송요금 및 정책

Terms & Conditions

Intellectual Property Promise

도구

도구

무료 샘플 정책

Calculator Application

Scientific Reviews

Topics

Product Guides

Blogs

Protocols

Brochures

Promotions

Events and Webinars

Genes

Biomedical Dictionary

Subscribe to our E-newsletter

Sorry, but the email address you supplied was invalid.

Thanks, your subscription has been confirmed. You will hear from us soon.

Submission failed, please try again later.

제품은 연구용 화학 시약이며 사람에게 사용할 수 없습니다. 환자에게는 판매하지 않습니다.

Copyright © 2013-2026 MedChemExpress. All Rights Reserved.

Site Map | Privacy and Cookie Policy

Online Service Online Customer Service

Contact Us

Happy to help!

MedChemExpress

Tel: 609-228-6898

E-mail: [email protected]

Technical Support: [email protected]

MedChemExpress

We use cookies

MedChemExpress values your privacy and your trust is important to us. We use cookies to enhance your website experience. Some cookies are necessary to run the website. Privacy and Cookie Policy

UK140

Biological Activity

제품 설명

IC50 & Target

Chemical Information

순도&문서

References

Calculators

Help & FAQs

UK140 Related Classifications

HY-P10878 Related Classifications

Bioz

Keywords

Your Recently Viewed Products

IC₅₀ & Target