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Cat. No.: HY-118904

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VL-0395

VL-0395 is a CCK1 selective antagonist with IC₅₀ of 0.197 μM for CCK1 in rat pancreatic acinar cells.

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CAS No.: 620167-11-5
화학식: C₂₅H₂₁N₃O₄
분자량:427.45

보관:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (274 KB)

VL-0395 Chemical Structure

CAS No.: 620167-11-5

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- 제품 설명
- Cellular Effect
Chemical Information
순도&문서
References
Calculators
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Bioz

Biological Activity

제품 설명

VL-0395 is a CCK1 selective antagonist with IC₅₀ of 0.197 μM for CCK1 in rat pancreatic acinar cells^[1].

All Cholecystokinin Receptor Isoforms :

CCKAR
CCKBR

Cellular Effect

Cell Line	Type	Value	Description	References
A-431	IC₅₀	197 nM Compound: VL-0395	Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor in A431 cells Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor in A431 cells	[PMID: 16610788]

Chemical Information

CAS No. 620167-11-5
분자량 427.45
화학식 C₂₅H₂₁N₃O₄
SMILES

O=C(C(CC1=CC=CC=C1)NC(C2=C(NC(C3=CC4=C(N3)C=CC=C4)=O)C=CC=C2)=O)O
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.

순도&문서

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (274 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Varnavas A, et al. Anthranilic acid based CCK1 receptor antagonists: preliminary investigation on their second “touch point”[J]. European journal of medicinal chemistry, 2005, 40(6): 563-581. [Content Brief]

Calculators

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
- 제품 설명
Chemical Information
순도&문서
References

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VL-0395

All Cholecystokinin Receptor Isoforms

Biological Activity

Chemical Information

순도&문서

References

Calculators

Help & FAQs

VL-0395 Related Classifications

HY-118904 Related Classifications