lucPpy-IN-1
Based on 1 Customer Validation
lucPpy-IN-1 (compound 9) is an ATP-dependent luciferase from Photinus pyralis (lucPpy) inhibitor with an IC50 value of 4.0 μM. lucPpy-IN-1 can be used for the research of target’s agentgability.
For research use only. We do not sell to patients.
- Purity: 99.48%
- CAS No.: 546100-66-7
- Formula: C25H23N5O
- Molecular Weight:409.48
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Storage:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
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Biological Activity
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Chemical Information
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Solvent & Solubility
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
IC50: 4.0 µM (lucPpy)[1]
lucPpy-IN-1 (0.1 nM-100 μM) inhibits activity of lucPpy with an IC50 value of 4.0 μM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 546100-66-7
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Appearance Solid
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Molecular Weight 409.48
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Formula C25H23N5O
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Color Pink to orange
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SMILES
O=C(C1=CC(C2=CC=C(C)C=C2)=NC3=CC=CC=C13)N4CCN(C5=NC=CC=N5)CC4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : 125 mg/mL (305.27 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (273 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.4421 mL | 12.2106 mL | 24.4212 mL | 61.0530 mL |
| 5 mM | 0.4884 mL | 2.4421 mL | 4.8842 mL | 12.2106 mL | |
| 10 mM | 0.2442 mL | 1.2211 mL | 2.4421 mL | 6.1053 mL | |
| 15 mM | 0.1628 mL | 0.8140 mL | 1.6281 mL | 4.0702 mL | |
| 20 mM | 0.1221 mL | 0.6105 mL | 1.2211 mL | 3.0527 mL | |
| 25 mM | 0.0977 mL | 0.4884 mL | 0.9768 mL | 2.4421 mL | |
| 30 mM | 0.0814 mL | 0.4070 mL | 0.8140 mL | 2.0351 mL | |
| 40 mM | 0.0611 mL | 0.3053 mL | 0.6105 mL | 1.5263 mL | |
| 50 mM | 0.0488 mL | 0.2442 mL | 0.4884 mL | 1.2211 mL | |
| 60 mM | 0.0407 mL | 0.2035 mL | 0.4070 mL | 1.0176 mL | |
| 80 mM | 0.0305 mL | 0.1526 mL | 0.3053 mL | 0.7632 mL | |
| 100 mM | 0.0244 mL | 0.1221 mL | 0.2442 mL | 0.6105 mL |
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