P2X2R antagonist-1
P2X2R antagonist-1 (compound 66) is a P2X2 receptor antagonist derived from Reactive Blue 4 (HY-125815). P2X2R antagonist-1 shows high selectivity for P2X4, P2X7, P2Y2, P2Y4, P2Y6 and P2Y12 receptors, moderate selectivity for P2X1 and P2X3 receptors, and exhibits higher potency toward homomeric P2X2 receptors than heteromeric P2X2/3 receptors. P2X2R antagonist-1 competitively inhibits ATP-mediated currents. P2X2R antagonist-1 can be used in research related to pain and urinary incontinence.
For research use only. We do not sell to patients.
- CAS No.: 13112-05-5
- Formula: C23H14N6Na2O10S2
- Molecular Weight:644.50
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
- Purity & Documentation
- References
-
Help & FAQs
All P2X Receptor Isoforms
More
Biological Activity
|
P2X2 Receptor |
Chemical Information
-
CAS No. 13112-05-5
-
Molecular Weight 644.50
-
Formula C23H14N6Na2O10S2
-
SMILES
O=C1N=C(NC2=CC(NC(C=C(S(=O)(O[Na])=O)C(N)=C3C(C4=C5C=CC=C4)=O)=C3C5=O)=CC=C2S(=O)(O[Na])=O)NC(N1)=O
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
P2X2R antagonist-1 Related Classifications
HY-184044 Related Classifications
Powered by Bioz