P2X4 antagonist-2
P2X4 antagonist-2 is an antagonist for P2X4 with an IC50 of 24 nM.
For research use only. We do not sell to patients.
- CAS No.: 2055601-24-4
- Formula: C21H16ClF3N2O4S
- Molecular Weight:484.88
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All P2X Receptor Isoforms
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Biological Activity
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P2X4 Receptor 24 nM (IC50) |
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Cell Line
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Type | Value | Description | References |
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| HEK293 | IC50 |
24 nM
Compound: 21
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Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins and measured every 2 secs for 120 secs by Fluo8-AM staining based FLIPR assay
Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins and measured every 2 secs for 120 secs by Fluo8-AM staining based FLIPR assay
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[PMID: 31746599] |
Chemical Information
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CAS No. 2055601-24-4
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Molecular Weight 484.88
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Formula C21H16ClF3N2O4S
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SMILES
O=C(CC1=C(C(F)(F)F)C=CC=C1)NC2=CC=C(C(S(=O)(N)=O)=C2)OC3=CC(Cl)=CC=C3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
P2X4 antagonist-2 Related Classifications
HY-160677 Related Classifications
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