PAT-IN-1
PAT-IN-1 is a protein acyl transferases (PAT) inhibitor. PAT-IN-1 competitively inhibits Erf2 autopalmitoylation (WO2017011518A1; compound 13).
For research use only. We do not sell to patients.
- CAS No.: 2066571-97-7
- Formula: C45H68N4O
- Molecular Weight:681.05
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
PAT-IN-1 (compound 13) completely inhibits growth of RJY1941 (control) at 20 μΜ, but has no detectable effect at lower concentrations. PAT-IN-1 inhibits (100%) the growth of RJY1942 (palmitoylation sensitive) at 5 μΜ[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2066571-97-7
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Molecular Weight 681.05
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Formula C45H68N4O
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SMILES
CC(C1=CC=C(C=C1)CC(C)C)CN(CCN(C2)CCCC[C@@H]3N(CCNC3)CC(C4=CC=C(C=C4)CC(C)C)C)[C@H]2CC5=CC=C(C=C5)O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)