1. GPCR/G Protein Neuronal Signaling
  2. Adrenergic Receptor
  3. Piperoxan

Piperoxan is an α1-adrenergic receptor antagonist. Piperoxan exhibits a Ki value of 360 nM for inhibiting 3H-prazosin binding to rat brain α1-adrenoceptors. Piperoxan can be used for the research of adrenergic system-related diseases.

For research use only. We do not sell to patients.

Piperoxan

Piperoxan Chemical Structure

CAS No. : 59-39-2

Size Stock
50 mg   Get quote  
100 mg   Get quote  
250 mg   Get quote  

* Please select Quantity before adding items.

This product is a controlled substance and not for sale in your territory.

Other In-stock Forms of Piperoxan:

Other Forms of Piperoxan:

Top Publications Citing Use of Products

View All Adrenergic Receptor Isoform Specific Products:

  • Biological Activity

  • Purity & Documentation

  • References

  • Customer Review

Description

Piperoxan is an α1-adrenergic receptor antagonist. Piperoxan exhibits a Ki value of 360 nM for inhibiting 3H-prazosin binding to rat brain α1-adrenoceptors. Piperoxan can be used for the research of adrenergic system-related diseases[1].

IC50 & Target[1]

rat α1-adrenergic receptor

360 nM (Ki)

In Vitro

Piperoxan (30 min) inhibits specific 3H-prazosin binding to rat brain minus cerebella membranes with a Ki of 360 nM, indicating moderate affinity for the α1-adrenergic receptor population labelled by 3H-prazosin[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

233.31

Formula

C14H19NO2

CAS No.
SMILES

O1C=2C=CC=CC2OC(C1)CN3CCCCC3

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
  • No file chosen (Maximum size is: 1024 Kb)
  • If you have published this work, please enter the PubMed ID.
  • Your name will appear on the site.
  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Your Recently Viewed Products:

Inquiry Online

Your information is safe with us. * Required Fields.

Product Name

 

Requested Quantity *

Applicant Name *

 

Salutation

Email Address *

 

Phone Number *

Department

 

Organization Name *

City

State

Country or Region *

     

Remarks

Bulk Inquiry

Inquiry Information

Product Name:
Piperoxan
Cat. No.:
HY-W556123
Quantity:
MCE Japan Authorized Agent: