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Cat. No.: HY-17037AS

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Pirenzepine-d₁₁

(Synonyms: LS 519 free base-d11; Pirenzepin-d11; Gastrozepin-d11)

Pirenzepine-d₁₁ (LS 519 (free base)-d₁₁; Pirenzepin-d₁₁; Gastrozepin-d₁₁) is the deuterium labeled Pirenzepine (HY-17037A). Pirenzepine (LS 519 free base) is a selective M1 mAChR (muscarinic acetylcholine receptor) antagonist. Pirenzepine reduces gastric acid secretion and reduces muscle spasm, can be used in peptic ulcers research. Pirenzepine shows anti-proliferative activity to cancer cells.

For research use only. We do not sell to patients.

Formula: C₁₉H₁₀D₁₁N₅O₂
Molecular Weight:362.47

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (247 KB)

Pirenzepine-d₁₁ Chemical Structure

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Biological Activity
- Description
- In Vitro
- Application
Chemical Information
Purity & Documentation
Calculators
Help & FAQs
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Biological Activity

Description

All mAChR Isoforms :

In Vitro

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Application

1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.

Chemical Information

Unlabeled Cas 28797-61-7
Molecular Weight 362.47
Formula C₁₉H₁₀D₁₁N₅O₂
SMILES

O=C(N(C1=C2C=CC=C1)C3=C(C=CC=N3)NC2=O)CN4C([2H])(C([2H])(N(C([2H])(C4([2H])[2H])[2H])C([2H])([2H])[2H])[2H])[2H]
Synonyms

LS 519 free base-d11; Pirenzepin-d11; Gastrozepin-d11
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.