PSI-112
PSI-112 is a YO-class μPlm inhibitor, with IC50 values of 0.38 μM, 1.48 μM and 0.37 μM against the wild-type, F587A mutant and K607A mutant, respectively. PSI-112 shows low affinity for uPA. PSI-112 can be used in cancer research.
For research use only. We do not sell to patients.
- CAS No.: 1854997-77-5
- Formula: C35H48N4O3
- Molecular Weight:572.78
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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μPlm 0.38 μM (IC50) |
PSI-112 inhibits wild-type μPlm with an IC50 of 0.38 μM, and its affinity for uPA (IC50 >25 μM) is lower than that for μPlm[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 1854997-77-5
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Molecular Weight 572.78
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Formula C35H48N4O3
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SMILES
O=C([C@@H]1CC[C@H](CC1)CN)N[C@H](C(NCCCCCCCC)=O)CC(C=C2)=CC=C2OCC3=NC4=C(C=CC=C4)C=C3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
PSI-112 Related Classifications
HY-182565 Related Classifications
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