Development of TRPM8 Antagonists to Treat Chronic Pain and Migraine

  • Pharmaceuticals (Basel). 2017 Mar 30;10(2):37. doi: 10.3390/ph10020037.
Andy D Weyer  1 Sonya G Lehto  2
Affiliations
Abstract

A review. Development of pharmaceutical antagonists of transient receptor potential melastatin 8 (TRPM8) have been pursued for the treatment of chronic pain and migraine. This review focuses on the current state of this progress.

Keywords
cold analgesia; cold hyperalgesia; mechanical hyperalgesia; menthol; migraine; pain; transient receptor potential melastatin 8 (TRPM*).
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