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Cat. No.: HY-177347

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RSK2-IN-6

RSK2-IN-5 (compoud C2) is a p90 ribosomal S6 kinase 2 (RSK2) inhibitor with a K_d of 856 nM. RSK2-IN-5 exhibits antitumor activity against breast cancer and melanoma cancer cells.

For research use only. We do not sell to patients.

CAS No.: 304474-86-0
Formula: C₁₇H₁₅N₅O₃S
Molecular Weight:369.40

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (274 KB)

RSK2-IN-6 Chemical Structure

CAS No.: 304474-86-0

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Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

RSK2-IN-5 (compoud C2) is a p90 ribosomal S6 kinase 2 (RSK2) inhibitor with a K_d of 856 nM. RSK2-IN-5 exhibits antitumor activity against breast cancer and melanoma cancer cells^[1].

All Ribosomal S6 Kinase (RSK) Isoforms :

Chemical Information

CAS No. 304474-86-0
Molecular Weight 369.40
Formula C₁₇H₁₅N₅O₃S
SMILES

O=C(C1=CC=CC([N+]([O-])=O)=C1)NNC2=C3C(CCCC4)=C4SC3=NC=N2
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (274 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Yue Zhao, et al. Discovery of novel p90 ribosomal S6 kinase 2 inhibitors for potential cancer treatment through ligand-based and structure-based virtual screening methods. Chemometrics and Intelligent Laboratory Systems. Volume 217, 15 October 2021, 104402

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

100 mg

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