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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
17 Results for "
CREBBP
" in MedChemExpress (MCE) Product Catalog:
Products (17)
17 Results for "CREBBP" in MCE Product Catalog:
Target:
Research Areas:
CBP/p300-IN-10 is a highly potent histone acetyltransferase EP300 and CREBBP with IC50 values of 26 nM and 39 nM, respectively. CBP/p300-IN-10 can be used to research anticancer .
Cat. No.: HY-RS03155
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CREBBP Human Pre-designed siRNA Set A contains three designed siRNAs for CREBBP gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-116237
CAS No.: 1219576-50-7
Target:
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CREBBP-IN-9 (Compound 9) is an inhibitor for CREBBP with an Kd of 29 μM .
Cat. No.: HY-128362
CAS No.: 2259641-24-0
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Ep300/CREBBP-IN-8 (Example 37) is a potent and orally active Ep300 and CREBBP inhibitor with IC50s of 0.014 and 0.018 μM, respectively. Ep300/CREBBP-IN-8 can be used for the research of cancer .
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OXFBD04 is a potent and selective BRD4 inhibitor with an IC50 of 166 nM. OXFBD04 is a potent BET bromodomain ligand with additional modest affinity for the CREBBP bromodomain. OXFBD04 has anti-cancer activity .
Cat. No.: HY-114971
CAS No.: 1801324-41-3
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Research Areas:
CREBBP-IN-1 (Compound 10) exhibits good affinity with CREBBP bromodomain with Kd of 0.77 μM .
Cat. No.: HY-128364
CAS No.: 2259641-47-7
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Ep300/CREBBP-IN-3 (Example 61) is a potent Ep300 and CREBBP inhibitor with IC50s of 0.056 and 0.095 μM, respectively. Ep300/CREBBP-IN-3 can be used for the research of cancer .
Cat. No.: HY-128367
CAS No.: 2259641-42-2
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Research Areas:
Ep300/CREBBP-IN-4 (Example 56) is a potent Ep300 and CREBBP inhibitor with IC50s of 0.024 and 0.064 μM, respectively. Ep300/CREBBP-IN-4 can be used for the research of cancer .
Cat. No.: HY-128363
CAS No.: 2259641-59-1
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Research Areas:
Ep300/CREBBP-IN-2 (Example 73) is a potent and orally active Ep300 and CREBBP inhibitor with IC50s of 0.052 and 0.148 μM, respectively. Ep300/CREBBP-IN-2 can be used for the research of cancer .
Cat. No.: HY-RS03156
Target:
Research Areas:
Crebbp Mouse Pre-designed siRNA Set A contains three designed siRNAs for Crebbp gene (Mouse), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS03157
Target:
Research Areas:
Crebbp Rat Pre-designed siRNA Set A contains three designed siRNAs for Crebbp gene (Rat), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-P702890
Purity: ≥ 90%, as determined by reducing SDS-PAGE.
Synonyms: CBP; KAT3A
Cat. No.: HY-P702891
Purity: ≥ 80%, as determined by reducing SDS-PAGE.
Synonyms: CBP; KAT3A
Cat. No.: HY-P702959
Purity: ≥ 90%, as determined by reducing SDS-PAGE.
Synonyms: CBP; KAT3A
Cat. No.: HY-122081
CAS No.: 1904647-34-2
Research Areas:
CPI-644 is a selective EP300/CBP bromodomain inhibitor, with an IC50 of 0.18 µM against the CBP bromodomain. CPI-644 reduces the proportion of FOXP3 + cells and downregulates the expression of LAG-3, CTLA-4 and PD-1. CPI-644 can be used in cancer-related research .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
