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Cat. No.: HY-116237

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CREBBP-IN-9

CREBBP-IN-9 (Compound 9) is an inhibitor for CREBBP with an K_d of 29 μM.

For research use only. We do not sell to patients.

CAS No.: 1219576-50-7
Formula: C₁₆H₁₅N₅O₂S
Molecular Weight:341.39

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (269 KB)

CREBBP-IN-9 Chemical Structure

CAS No.: 1219576-50-7

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Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

CREBBP-IN-9 (Compound 9) is an inhibitor for CREBBP with an K_d of 29 μM^[1].

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Chemical Information

CAS No. 1219576-50-7
Molecular Weight 341.39
Formula C₁₆H₁₅N₅O₂S
SMILES

O=C(NC1=CC=CC(C(C)=O)=C1)C2=C(SC(C)=C2C)N3N=NN=C3
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (269 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Xu M, et al., Discovery of CREBBP Bromodomain Inhibitors by High-Throughput Docking and Hit Optimization Guided by Molecular Dynamics. J Med Chem. 2016 Feb 25;59(4):1340-9. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

100 mg

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