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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
23 Results for "
SST1
" in MedChemExpress (MCE) Product Catalog:
Products (23)
23 Results for "SST1" in MCE Product Catalog:
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6 Publications Verification
Cat. No.: HY-79135
Synonyms: SOM230 ditrifluoroacetate; Pasireotide TFA salt
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Pasireotide (SOM230) ditrifluoroacetate, a long-acting cyclohexapeptide somatostatin analogue, can improve agonist activity at somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9, respectively). Pasireotide ditrifluoroacetate exhibits antisecretory, antiproliferative, and proapoptotic activity [1] .
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3
3 Cited Publications
Cat. No.: HY-P1202
CAS No.: 183658-72-2
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3
3 Cited Publications
Cat. No.: HY-P1202A
CAS No.: 2828432-46-6
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2
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1
1 Cited Publications
Cat. No.: HY-P1932
CAS No.: 186901-48-4
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1
1 Cited Publications
Cat. No.: HY-P1206
CAS No.: 174688-78-9
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1
1 Cited Publications
Cat. No.: HY-P1932A
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Cat. No.: HY-111615
CAS No.: 848647-56-3
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SRA880 is a non-peptide and selective somatostatin sst(1) receptor antagonist. SRA880 exhibits antidepressant-like effects when in combination with Imipramine (HY-B1490A) [1].
Cat. No.: HY-177282
CAS No.: 524743-70-2
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Cardiovascular Disease Neurological Disease Inflammation/Immunology Cancer
SST1 receptor antagonist-2 (Example 2) is a piperazine derivative and a somatostatin receptor 1 (SST1) antagonist. SST1 receptor antagonist-2 can be used in the research of psychiatric diseases, neurodegenerative diseases, tumors, as well as vascular disorders and immunological diseases [1].
Cat. No.: HY-177278
CAS No.: 868057-23-2
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SST1 receptor antagonist-1 (Compound 23) is a selective Somatostatin receptor 1 (SST1) antagonist with pKds of 9.11 and 8.79 for rSST1 and hSST1, respectively. SST1 receptor antagonist-1 can be used for retinal and endocrine dysfunctions, cancer and neuropsychiatric disorders research [1].
Cat. No.: HY-P4469
CAS No.: 341519-04-8
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Cat. No.: HY-125382
CAS No.: 217480-24-5
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L-797591 is a selective sst1 agonist. L-797591 mimicks the effects of SRIF-14 and SRIF-28 by potently inhibiting either Forskolin (HY-15371)-stimulated or CRH-stimulated cAMP accumulation [1].
Cat. No.: HY-16381B
CAS No.: 1421446-02-7
Synonyms: SOM230 (diaspartate)
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Pasireotide (SOM230) diaspartate, a long-acting cyclohexapeptide somatostatin analogue, can improve agonist activity at somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9, respectively). Pasireotide diaspartate exhibits antisecretory, antiproliferative, and proapoptotic activity [1] .
Cat. No.: HY-125382A
CAS No.: 3026641-74-4
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L-797591 hydrochloride is a selective sst1 agonist. L-797591 hydrochloride mimicks the effects of SRIF-14 and SRIF-28 by potently inhibiting either Forskolin (HY-15371)-stimulated or CRH-stimulated cAMP accumulation [1].
Cat. No.: HY-175053
Synonyms: SOM230 (aspartate) TFA
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
