1. GPCR/G Protein
  2. Somatostatin Receptor
  3. CYN 154806 TFA

CYN 154806 TFA 

Cat. No.: HY-P1202A Purity: 99.97%
Handling Instructions

CYN 154806 (TFA), a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively.

For research use only. We do not sell to patients.

Custom Peptide Synthesis

CYN 154806 TFA Chemical Structure

CYN 154806 TFA Chemical Structure

Size Price Stock Quantity
10 mM * 1 mL in Water USD 1414 In-stock
Estimated Time of Arrival: December 31
1 mg USD 180 In-stock
Estimated Time of Arrival: December 31
5 mg USD 580 In-stock
Estimated Time of Arrival: December 31
10 mg USD 980 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
100 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

Based on 1 publication(s) in Google Scholar

Other Forms of CYN 154806 TFA:

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  • Biological Activity

  • Technical Information

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Description

CYN 154806 (TFA), a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively[1][2].

IC50 & Target

Somatostatin Receptor[1].

Storage
Powder -80°C 2 years
  -20°C 1 year
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

H2O : 50 mg/mL (38.13 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 0.7626 mL 3.8128 mL 7.6257 mL
5 mM 0.1525 mL 0.7626 mL 1.5251 mL
10 mM 0.0763 mL 0.3813 mL 0.7626 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

1311.36

Formula

C₅₈H₆₉F₃N₁₂O₁₆S₂

Sequence

Ac-FCYWKTCY-NH2 (Disulfide bridge: Cys2-Cys7)

Sequence Shortening

Ac-Phe-Cys-Tyr-Trp-Lys-Thr-Cys-Tyr-NH2 (Disulfide bridge: Cys2-Cys7)

Shipping

Room temperature in continental US; may vary elsewhere

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
CYN 154806 TFA
Cat. No.:
HY-P1202A
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CYN 154806 TFA

Cat. No.: HY-P1202A