TMPBM ligand-1
TMPBM ligand-1 (compound d9A1 warhead) is an SLC9A1 ligand. TMPBM ligand-1 can be used for the synthesis of d9A1-2 (HY-183892). TMPBM ligand-1 is applicable to research on cancers such as chronic myeloid leukemia.
For research use only. We do not sell to patients.
- CAS No.: 2640254-08-4
- Formula: C23H24FN3O2
- Molecular Weight:393.45
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Description
IC50 & Target
[1]|
SLC9A1 |
In Vitro
PROTACs contain two different ligands connected by a linker; one is a ligand for an E3 ubiquitin ligase and the other is for the target protein. PROTACs exploit the intracellular ubiquitin-proteasome system to selectively degrade target proteins.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2640254-08-4
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Molecular Weight 393.45
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Formula C23H24FN3O2
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SMILES
O=C(O)C1=CC=C(C2=CC=C(F)C(C)=C2)C(N3CCC(C4=C(C)N=CN4)CC3)=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)